反向激动剂指一种新分类概念。
摘要反向激动剂指一种新分类概念。
与阻断激动剂效应的拮抗剂不同，反向激动剂产生的效应与激动剂相反。
Different form antagonist that blocks the effect of agonist, inverse agonist produces opposite effect to that of agonist.
本发明提供了具有胰高血糖素受体拮抗剂活性或反向激动剂活性的、新颖的式i化合物及其药学上可接受的盐和共晶体。
The present invention provides for novel compounds of Formula (I) and pharmaceutically acceptable salts and co-crystals thereof which have glucagon receptor antagonist or inverse agonist activity.
本发明提供了具有胰高血糖素受体拮抗剂活性或反向激动剂活性的、新颖的式i化合物及其药学上可接受的盐和共晶体。
The present invention provides for novel compounds of Formula (I) and pharmaceutically acceptable salts and co-crystals thereof which have glucagon receptor antagonist or inverse agonist activity.
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