反向激动剂指一种新分类概念。
摘要反向激动剂指一种新分类概念。
2受体激动剂的镇静效果机理是什么?。
受体激动剂是兽药的一种。
小剂量左旋多巴和多巴胺激动剂治疗有效。
Low dose levodopa and dopamine agonists are effective in controlling most symptoms of the disorder.
一优选调节物为激动剂。
目的：探讨钾通道激动剂在哮喘防治中的作用。
Objective: to study the role of potassium channel activator in treatment of asthma.
非竞争性拮抗剂可阻止激动剂在特定受体部位产生任何效应。
A noncompetitive antagonist prevents the agonist from producing any effect at a given receptor site.
结果：药理评价显示甲磺酸培高利特是一典型D受体激动剂。
RESULTS:Pharmacological evaluation showed that Pergolide mesylate is a specific dopminergic DA receptor agonist.
哮喘病人外周血白细胞受激动剂作用会产生更大的细胞反应。
Greater leukocyte reaction is induced by agonist in patient with asthma.
目的研究兴奋性氨基酸受体激动剂对雌性大鼠青春期启动的影响。
Objective to observe the effect of excitatory amino acids receptor agonist on the onset of puberty in female rats.
目的：探讨腺苷a1受体激动剂延迟预处理对大鼠心脏的保护效果。
Objective: to study the protecting effect of delayed preconditioning with A1 selective adenosine receptor agonist in donor heart preservation.
与阻断激动剂效应的拮抗剂不同，反向激动剂产生的效应与激动剂相反。
Different form antagonist that blocks the effect of agonist, inverse agonist produces opposite effect to that of agonist.
而以tlr - 4激动剂LPS处理的滋养层细胞并未有细胞活性下降。
Treatment of cells with the TLR-4 agonist, LPS, did not reduce trophoblast cell viability.
结果表明，GABA受体激动剂可提高大鼠痛阈，而拮抗剂降低大鼠痛阈。
The results showed that GABA receptor agonists increased rat's pt, and GABA receptor antagonists decreased pt.
目前世界药物市场上有三分之一的小分子药物是GPCR的激动剂和拮抗剂。
So far, one third of approved small molecular drugs sold in market are the agonists or antagonists of GPCR.
患者可选用其它治疗药物，包括三种与心脏瓣膜疾病无关的其它多巴胺激动剂。
There are alternative therapies available for Parkinson's disease, including three other dopamine agonists that have not been associated with valvular heart disease.
百泌达是FDA批准的治疗2型糖尿病的首个GLP- 1受体激动剂药物。
BYETTA is the first FDA-approved GLP-1 receptor agonist for the treatment of type 2 diabetes.
目的：对比分析多巴胺1受体激动剂非诺多泮对兔肺动脉和肠系膜动脉的影响。
Objective: To evaluate and compare the effects of DA 1 receptor agonist, fenoldopam, rabbit pulmonary and mesenteric arteries.
目的研究多巴胺受体激动剂对乙醇引起大鼠纹状体抗坏血酸(AA)释放的影响。
AIM to study the effects of dopamine receptor agonists on ethanol induced striatal ascorbic acid (AA) release in rats.
目的研究M3受体激动剂毛果芸香碱对离体大鼠心肌缺血再灌注损伤的保护作用。
OBJECTIVE To investigate the protective effects of M3 receptor agonist pilocarpine on myocardial ischemia-reperfusion injury in isolated rat hearts.
然而，大多数临床试验这些激动剂都是单独使用的，没有显示出其治疗癌症的效应。
However, most clinical trials conducted with these agonists as monotherapy in patients with cancer have not shown a benefit.
CCK受体激动剂与拮抗剂的研究深入，促进了人们对CCK生理功能的深入认识。
With study development of CCK receptor antagonist and agonist, people have deep understanding about CCK's physiological function.
目前的研究目的是评估使用多巴胺激动剂治疗的泌乳素瘤病人瓣膜性心脏病的患病率。
The aim of the present study was to assess the prevalence of valvular heart disease in patients treated with dopamine agonists for prolactinomas.
因而寻找选择性5 - HT _ (2c)受体激动剂成为一个药物研究及开发的热点。
So searching selective 5-ht_ (2c) receptor agonists has become a focus in drug research and development.
通过烟碱乙酰胆碱受体7激动剂阻断细胞因子生成是在炎症发生前治疗中风的一种新疗法。
Blockade of cytokine production by 7 nicotinic acetylcholine receptor agonists is a novel therapeutic option to treat stroke in a proinflammatory context.
体外研究的资料指出多巴受体激动剂有抗氧化，清除自由基的性质，可能有一定的神经保护效应。
In vitro results suggest that dopamine agonists may have the potential neuroprotective effect because of the properties of antioxidation and scavenging radical oxygen.
结论：GLP - 1受体激动剂治疗后的体重减轻与心血管危险因素谱向更有益的方向转变有关。
CONCLUSIONS Weight reduction with GLP-1 receptor agonists was associated with a shift toward a more favorable cardiovascular risk profile.
目的：使用麦角衍生的多巴胺激动剂，已经证实帕金森病人使用培高利特和卡麦角林可能增加瓣膜心脏病。
Objective: Treatment with ergot-derived dopamine agonists, pergolide, and cabergoline has been associated with an increased frequency of valvular heart disease in Parkinson's disease.
目的：使用麦角衍生的多巴胺激动剂，已经证实帕金森病人使用培高利特和卡麦角林可能增加瓣膜心脏病。
Objective: Treatment with ergot-derived dopamine agonists, pergolide, and cabergoline has been associated with an increased frequency of valvular heart disease in Parkinson's disease.
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