受体激动剂是兽药的一种。
2受体激动剂的镇静效果机理是什么?。
结果:药理评价显示甲磺酸培高利特是一典型D受体激动剂。
RESULTS:Pharmacological evaluation showed that Pergolide mesylate is a specific dopminergic DA receptor agonist.
本文提供了反转或阻止靶细胞对死亡受体激动剂的抗性的方法。
Provided herein is a method of reversing or preventing a target cell's resistance to a death receptor agonist.
目的研究兴奋性氨基酸受体激动剂对雌性大鼠青春期启动的影响。
Objective to observe the effect of excitatory amino acids receptor agonist on the onset of puberty in female rats.
目的:探讨腺苷a1受体激动剂延迟预处理对大鼠心脏的保护效果。
Objective: to study the protecting effect of delayed preconditioning with A1 selective adenosine receptor agonist in donor heart preservation.
结果表明,GABA受体激动剂可提高大鼠痛阈,而拮抗剂降低大鼠痛阈。
The results showed that GABA receptor agonists increased rat's pt, and GABA receptor antagonists decreased pt.
本发明公开了一种重组PAC1受体激动剂rmmax及其表达方法与应用。
The invention discloses a recomposing PAC1 receptor excitant RMMAX and an expressing method and application thereof.
百泌达是FDA批准的治疗2型糖尿病的首个GLP- 1受体激动剂药物。
BYETTA is the first FDA-approved GLP-1 receptor agonist for the treatment of type 2 diabetes.
目的:对比分析多巴胺1受体激动剂非诺多泮对兔肺动脉和肠系膜动脉的影响。
Objective: To evaluate and compare the effects of DA 1 receptor agonist, fenoldopam, rabbit pulmonary and mesenteric arteries.
目的研究多巴胺受体激动剂对乙醇引起大鼠纹状体抗坏血酸(AA)释放的影响。
AIM to study the effects of dopamine receptor agonists on ethanol induced striatal ascorbic acid (AA) release in rats.
目的研究M3受体激动剂毛果芸香碱对离体大鼠心肌缺血再灌注损伤的保护作用。
OBJECTIVE To investigate the protective effects of M3 receptor agonist pilocarpine on myocardial ischemia-reperfusion injury in isolated rat hearts.
结论京尼平苷具有与GLP - 1受体激动剂类似的神经营养和神经保护功能。
CONCLUSION Geniposide has the similar function as the agonist for GLP-1 receptor, including neurotrophic and neuroprotective effects.
CCK受体激动剂与拮抗剂的研究深入,促进了人们对CCK生理功能的深入认识。
With study development of CCK receptor antagonist and agonist, people have deep understanding about CCK's physiological function.
因而寻找选择性5 - HT _ (2c)受体激动剂成为一个药物研究及开发的热点。
So searching selective 5-ht_ (2c) receptor agonists has become a focus in drug research and development.
利拉鲁肽是一种GLP - 1受体激动剂,这类药可在用餐后促使胰腺分泌更多的胰岛素。
Victoza is in a class of medicines known as glucagon-like peptide-1 (GLP-1) receptor agonists that help the pancreas make more insulin after eating a meal.
如果我们能够研发出“更聪明的药物”,比如瘦素受体激动剂,那么它肯定有巨大的治疗潜力。
If you could get a clever leptin agonist molecule then there is of course huge potential for the treatment.
体外研究的资料指出多巴受体激动剂有抗氧化,清除自由基的性质,可能有一定的神经保护效应。
In vitro results suggest that dopamine agonists may have the potential neuroprotective effect because of the properties of antioxidation and scavenging radical oxygen.
结论:GLP - 1受体激动剂治疗后的体重减轻与心血管危险因素谱向更有益的方向转变有关。
CONCLUSIONS Weight reduction with GLP-1 receptor agonists was associated with a shift toward a more favorable cardiovascular risk profile.
肠易激综合症5 - HT 3受体拮抗剂和5羟色胺受体激动剂的疗效:系统性回顾和荟萃分析。
Efficacy of 5-ht3 antagonists and 5-ht4 agonists in irritable bowel syndrome: systematic review and meta-analysis.
研究人员先前报道应用β-肾上腺素能受体激动剂治疗的疾病与小腿静脉溃疡之间有不可解释的相关性。
The researchers previously reported "unexplainable associations" between diseases treated with beta-adrenergic agents and the onset of a venous leg ulcer.
BYDUREON和百泌达(BYETTA)都属于胰高血糖素样肽(GLP - 1)受体激动剂类药物。
BYDUREON and BYETTA belong to the glucagon-like peptide-1 (GLP-1) receptor agonist class of medications.
而类胰蛋白酶受体激动剂对肥大细胞类胰蛋白酶分泌的促进作用则表明类胰蛋白酶是肥大细胞激活的正反馈性刺激剂。
Stimulation of tryptase release from mast cells by tryptase receptor agonists indicated that tryptase can stimulate mast cells in a positive feedback way.
我们通过本研究探讨了新型的D3受体激动剂普拉克索和罗匹尼罗对神经营养因子的调节作用和其对DA神经元的保护作用。
The present study discussed that the new D3 receptor agonists, pramipexole and ropinirole, mediate neurotrophic effects on DA neurons in fetal rat ventral mesencephalic cultures.
大量研究证据表明,5 - HT _ (2c)受体激动剂可能在治疗肥胖、焦虑、抑郁、强迫症和癫痫等疾病方面有疗效。
Strong evidences exist to support the use of 5-ht_ (2c) receptor agonists as pharmacological treatment of many diseases, including obesity, drug abuse, anxiety, depression, OCD and epilepsy.
因此,这项研究的目的就是比较增加ICS剂量与加入长效β-2受体激动剂两种方法在时间上对于控制哮喘疗效好坏的比较。
The goal of this post hoc analysis was to compare the effect of increasing the ICS dosage vs adding long-acting beta2-agonists on the time spent with well-controlled or poorly controlled asthma.
注射疗法,如GLP受体激动剂,通常在稍晚阶段开始使用此,大多数同意使用注射疗法的患者均已经用两种口服药物而未能使血糖达标。
Injectable therapies like a GLP receptor agonists usually come at a slightly later stage so most of the patients who are willing to agree to an injectable therapy have failed on two oral agents also.
方法建立稳定的GLP-1受体激动剂高通量筛选模型,从天然药物中筛选活性成分;在PC12细胞中验证GLP-1受体激动剂的功能及作用机制。
METHODS Natural products were collected to screen in the stable cell line of GLP-1 receptor, and the active component was identified in the PC12 cells.
方法建立稳定的GLP-1受体激动剂高通量筛选模型,从天然药物中筛选活性成分;在PC12细胞中验证GLP-1受体激动剂的功能及作用机制。
METHODS Natural products were collected to screen in the stable cell line of GLP-1 receptor, and the active component was identified in the PC12 cells.
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