英语:partial agonist。指药物与受体有较强的亲和力,仅有较弱的内在活性。
前言: 目的: 合成多巴胺D, 受体部分激动剂BP897。
Objective:To synthesize BP897, a dopamine D3 receptor partial agonist.
一些含羟基芳香族植物精油类化合物对美洲大蠊的毒理学研究表明它们是章鱼胺受体的部分激动剂或拮抗剂。
Eugenol, cinnamic alcohol, phenyl methyl alcohol and phenyl ethyl alcohol have shown to be potential antagonists or partial agonists to octopaminergic receptors in pharmacologic studies.
对alpha4beta2受体来说,既然伐伦克林仅是部分激动剂--不是完全激动剂,它对吸烟者和非吸烟者的作用是不同的,她说。
Since varenicline is only a partial agonist—not a full agonist—at the alpha4beta2 receptor site, it performs differently in smokers and nonsmokers, she said.
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